Compounded medications are not FDA approved. FDA does not review compounded medications for safety, effectiveness, or quality before they are marketed.

Research library

Pending medical review. These summaries reflect widely reported findings from foundational trials of FDA-approved semaglutide and tirzepatide products. The section is excluded from search indexing until a named medical reviewer confirms each summary and adds DOI, PMID, and ClinicalTrials.gov identifiers. No summary below applies to compounded formulations.

STEP 1

Product studied
semaglutide 2.4 mg weekly (Wegovy dose) — an FDA-approved product, not a compounded formulation
Design
Randomized, double-blind, placebo-controlled; ~1,960 adults with overweight or obesity without diabetes; 68 weeks
Headline finding
Mean weight loss of roughly 15% of body weight with semaglutide 2.4 mg plus lifestyle intervention versus ~2.4% with placebo; gastrointestinal effects were the most common adverse events.
Citations
DOI / PMID / NCT to be confirmed and added at medical review — identifiers are never printed from memory
Applicability
Results apply to the trialed FDA-approved product and doses; they do not establish outcomes for compounded, microdose, oral, ODT, or sublingual formulations.

SURMOUNT-1

Product studied
tirzepatide 5/10/15 mg weekly (Zepbound doses) — an FDA-approved product, not a compounded formulation
Design
Randomized, double-blind, placebo-controlled; ~2,540 adults with obesity without diabetes; 72 weeks
Headline finding
Dose-dependent mean weight loss reaching roughly 20–21% at the highest dose versus ~3% with placebo; gastrointestinal events most common, typically during dose escalation.
Citations
DOI / PMID / NCT to be confirmed and added at medical review — identifiers are never printed from memory
Applicability
Results apply to the trialed FDA-approved product and doses; they do not establish outcomes for compounded, microdose, oral, ODT, or sublingual formulations.

SELECT

Product studied
semaglutide 2.4 mg weekly — an FDA-approved product, not a compounded formulation
Design
Randomized, double-blind, placebo-controlled cardiovascular-outcomes trial; ~17,600 adults with established cardiovascular disease and overweight or obesity, without diabetes; multi-year follow-up
Headline finding
Approximately a 20% relative reduction in major adverse cardiovascular events (cardiovascular death, nonfatal MI, nonfatal stroke) versus placebo.
Citations
DOI / PMID / NCT to be confirmed and added at medical review — identifiers are never printed from memory
Applicability
Results apply to the trialed FDA-approved product and doses; they do not establish outcomes for compounded, microdose, oral, ODT, or sublingual formulations.

SURMOUNT-4

Product studied
tirzepatide, maximum tolerated dose — an FDA-approved product, not a compounded formulation
Design
Randomized-withdrawal design: open-label tirzepatide lead-in, then randomization to continued tirzepatide or placebo; 88 weeks total
Headline finding
Continuing tirzepatide produced further weight loss after the lead-in, while switching to placebo led to substantial regain of lost weight — central evidence on discontinuation and weight regain.
Citations
DOI / PMID / NCT to be confirmed and added at medical review — identifiers are never printed from memory
Applicability
Results apply to the trialed FDA-approved product and doses; they do not establish outcomes for compounded, microdose, oral, ODT, or sublingual formulations.

SURMOUNT-5

Product studied
tirzepatide vs semaglutide, head-to-head — an FDA-approved product, not a compounded formulation
Design
Randomized, open-label; adults with obesity without diabetes; 72 weeks; funded by Eli Lilly
Headline finding
Tirzepatide produced greater mean weight loss than semaglutide 2.4 mg (roughly 20% versus 14%), with broadly similar gastrointestinal adverse-event profiles; the open-label design and sponsor funding are relevant limitations.
Citations
DOI / PMID / NCT to be confirmed and added at medical review — identifiers are never printed from memory
Applicability
Results apply to the trialed FDA-approved product and doses; they do not establish outcomes for compounded, microdose, oral, ODT, or sublingual formulations.

Reported weight-loss outcomes across pivotal trials

Mean total body-weight reduction in pivotal obesity trials · FDA-approved products at studied doses · these figures do NOT transfer to compounded, microdose, oral, ODT, or sublingual formulations
STEP 1 — semaglutide 2.4mgSTEP 1 — semaglutide 2.4mg: 14.9% (68 weeks)14.9%SURMOUNT-1 — tirzepatide 15mgSURMOUNT-1 — tirzepatide 15mg: 20.9% (72 weeks)20.9%SURMOUNT-1 — tirzepatide 10mgSURMOUNT-1 — tirzepatide 10mg: 19.5% (72 weeks)19.5%SURMOUNT-5 — tirzepatide (h2h)SURMOUNT-5 — tirzepatide (h2h): 20.2% (72 weeks)20.2%SURMOUNT-5 — semaglutide (h2h)SURMOUNT-5 — semaglutide (h2h): 13.7% (72 weeks)13.7%

FDA-approved injectable products at studied doses. These outcomes do not transfer to compounded, microdose, or oral/sublingual formulations. Values pending citation confirmation at medical review.

View chart data as a table
Mean total body-weight reduction in pivotal obesity trials
Trial & productMean weight reductionDuration
STEP 1 — semaglutide 2.4mg14.9%68 weeks
SURMOUNT-1 — tirzepatide 15mg20.9%72 weeks
SURMOUNT-1 — tirzepatide 10mg19.5%72 weeks
SURMOUNT-5 — tirzepatide (h2h)20.2%72 weeks
SURMOUNT-5 — semaglutide (h2h)13.7%72 weeks

These are widely reported headline figures from the pivotal trials of the FDA-approved injectable products at their studied doses, shown for scientific context and pending medical-reviewer confirmation of each value with its DOI/PMID/NCT. They are not evidence for any compounded preparation, any sub-therapeutic "microdose," or any oral/sublingual route. Percentages are placebo-subtracted or total means as reported and will be finalized with citations at review.

Planned coverage

Remaining STEP and SURMOUNT trials; SUSTAIN and SURPASS diabetes programs; PIONEER and OASIS oral-semaglutide programs; FLOW, SUMMIT, SURMOUNT-OSA, and ESSENCE outcomes trials; discontinuation and weight-regain meta-analyses; body-composition, sarcopenia, and frailty evidence; compounded-product real-world studies with funding and design disclosures; and research-only pages for investigational agents (retatrutide, CagriSema, cagrilintide, orforglipron, survodutide, mazdutide, amycretin). Investigational agents receive no purchase, provider, ranking, compounding, or dosing content — retatrutide and cagrilintide are not FDA approved and are not lawfully available as compounded treatments.